Cyprodenate

Summary

Cyprodenate (Actebral) is a stimulant drug.[1] It was used for counteracting the effects of benzodiazepine tranquillizer drugs before the development of newer antidotes such as flumazenil.[2] It produces dimethylethanolamine as a metabolite.[citation needed]

Cyprodenate
Clinical data
AHFS/Drugs.comInternational Drug Names
ATC code
Identifiers
  • 2-dimethylaminoethyl 3-cyclohexylpropanoate
CAS Number
  • 15585-86-1 checkY
PubChem CID
  • 71875
ChemSpider
  • 64892 checkY
UNII
  • I44VIC13P8
KEGG
  • D07764 checkY
ChEMBL
  • ChEMBL2106590
CompTox Dashboard (EPA)
  • DTXSID70165978 Edit this at Wikidata
ECHA InfoCard100.036.025 Edit this at Wikidata
Chemical and physical data
FormulaC13H25NO2
Molar mass227.348 g·mol−1
3D model (JSmol)
  • Interactive image
  • CN(C)CCOC(=O)CCC1CCCCC1
  • InChI=1S/C13H25NO2/c1-14(2)10-11-16-13(15)9-8-12-6-4-3-5-7-12/h12H,3-11H2,1-2H3 checkY
  • Key:MPOYJPINNSIHAK-UHFFFAOYSA-N checkY
  (verify)

See also edit

References edit

  1. ^ Dormard Y, Levron JC, Le Fur JM (February 1975). "Pharmacokinetic study of maleate acid of 2-(N,N-dimethylaminoethanol-14C1)-cyclohexylpropionate (cyprodenate) and of N,N-dimethylaminoethanol-14C1 in animals". Arzneimittel-Forschung. 25 (2): 201–7. PMID 1173033.
  2. ^ Bobkov I, Morozov IS (October 1982). "[Correction of psychodepressive effects of benzodiazepine tranquilizers by administration of psychostimulants]". Biulleten' Eksperimental'noi Biologii I Meditsiny. 94 (10): 48–51. doi:10.1007/BF00827201. PMID 6129008. S2CID 19153614.