Isamoltane (CGP-361A) is a drug used in scientific research. It acts as an antagonist at the β-adrenergic, 5-HT1A, and 5-HT1B receptors.[1] It has about five times the potency for the 5-HT1B receptor (21 nmol/L) over the 5-HT1A receptor (112 nmol/L).[2] It has anxiolytic effects in rodents.[3]
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Formula | C16H22N2O2 |
Molar mass | 274.364 g·mol−1 |
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