RQ-00203078 is a drug which acts as a potent and selective blocker of the TRPM8 ion channel, which is the main receptor responsible for the sensation of cold. It was developed as a potential analgesic, and blocks the development of hyperalgesia following exposure to cold temperatures or chronic morphine administration.[1][2][3]
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Formula | C21H13ClF6N2O5S |
Molar mass | 554.84 g·mol−1 |
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